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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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AVPR1B
arginine vasopressin receptor 1B
Chromosome 1 · 1q32.1
NCBI Gene: 553Ensembl: ENSG00000198049.7HGNC: HGNC:896UniProt: P47901
50PubMed Papers
20Diseases
7Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Receptor
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
symbiont entry into host cellpositive regulation of inositol phosphate biosynthetic processpositive regulation of arachidonate secretionplasma membranediabetes insipidusenuresishemorrhagehepatorenal syndrome
✦AI Summary

AVPR1B (arginine vasopressin receptor 1B) is a G protein-coupled receptor primarily expressed in pituitary corticotropes that mediates arginine vasopressin (AVP) stimulation of ACTH release, thereby regulating the hypothalamic-pituitary-adrenal (HPA) axis under stress 1. The receptor activates phospholipase C signaling, increasing cytosolic calcium and inositol phosphate biosynthesis, while also promoting vasoconstriction and regulating blood pressure 2. Clinically, AVPR1B agonists function as vasopressors in critically ill patients with vasodilatory shock, though they have not significantly reduced mortality compared to standard agents like norepinephrine 3. Genetic variation in AVPR1B contributes to psychiatric vulnerability. Multiple polymorphisms associate with childhood-onset mood disorders, particularly in females, with the Lys65Asn variant showing strongest association 1. AVPR1B variants also correlate with bipolar disorder psychotic features and influence prosocial behavior in gene-environment and gene-gene interactions with clock genes 45. The gene has undergone natural selection in human populations, with evidence of balancing selection in African and European populations, suggesting adaptive significance potentially related to mood regulation 6. AVPR1B antagonists demonstrate antidepressant properties, implicating this receptor in HPA axis dysregulation underlying mood pathology.

Sources cited
1
AVPR1B is a vasopressin receptor involved in vasoconstriction through vasopressor therapy in shock
PMID: 31646370
2
AVPR1B mediates vasopressor effects; vasopressin acting on AVPR1B has not decreased 28-day mortality in clinical trials
PMID: 32820475
3
AVPR1B SNPs associate with childhood-onset mood disorders, particularly in females; receptor modulates HPA axis stress response
PMID: 17909131
4
AVPR1B gene polymorphisms influence prosocial behavior through interaction with clock gene variants
PMID: 25309987
5
AVPR1B polymorphism rs28536160 associates with psychotic features in bipolar disorder
PMID: 22341483
6
AVPR1B has undergone natural selection in human populations with evidence of balancing selection; involved in mood and anxiety disorders
PMID: 19486526
Disease Associationsⓘ20
diabetes insipidusOpen Targets
0.58Moderate
enuresisOpen Targets
0.56Moderate
hemorrhageOpen Targets
0.56Moderate
hepatorenal syndromeOpen Targets
0.53Moderate
Nasal congestionOpen Targets
0.53Moderate
Central diabetes insipidusOpen Targets
0.50Moderate
head injuryOpen Targets
0.46Moderate
septic shockOpen Targets
0.38Weak
SepsisOpen Targets
0.37Weak
hypertensionOpen Targets
0.37Weak
amnesiaOpen Targets
0.37Weak
PolyuriaOpen Targets
0.37Weak
Renal insufficiencyOpen Targets
0.37Weak
von Willebrand disease (hereditary or acquired)Open Targets
0.37Weak
cirrhosis of liverOpen Targets
0.33Weak
cardiac arrestOpen Targets
0.33Weak
ShockOpen Targets
0.31Weak
PainOpen Targets
0.27Weak
benign muscle neoplasmOpen Targets
0.26Weak
HyponatremiaOpen Targets
0.26Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets7
ARGIPRESSIN TANNATEPhase III
Vasopressin receptor agonist
DESMOPRESSINApproved
Vasopressin receptor agonist
DESMOPRESSIN ACETATEApproved
Vasopressin receptor agonist
LYPRESSINApproved
Vasopressin receptor agonist
amnesia
NELIVAPTANPhase II
Vasopressin V1b receptor antagonist
anxiety disorder
TERLIPRESSINApproved
Vasopressin V1 receptor binding agent
hypertension
VASOPRESSINApproved
Vasopressin receptor agonist
diabetes insipidus
Related Genes
GNA13Protein interaction99%GNAQProtein interaction97%POMCProtein interaction94%CRHR1Protein interaction93%CRHProtein interaction92%LINC02210-CRHR1Protein interaction91%
Tissue Expression6 tissues
Brain
100%
Bone Marrow
5%
Liver
0%
Heart
0%
Lung
0%
Ovary
0%
Gene Interaction Network
Click a node to explore
AVPR1BGNA13GNAQPOMCCRHR1CRHLINC02210-CRHR1
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt P47901
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.19LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.85 [0.62–1.19]
RankingsWhere AVPR1B stands among ~20K protein-coding genes
  • #8,776of 20,598
    Most Researched50
  • #319of 1,025
    FDA-Approved Drug Targets5
  • #12,536of 17,882
    Most Constrained (LOEUF)1.19
Genes detectedAVPR1B
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Vasopressor therapy in critically ill patients with shock.
PMID: 31646370
Intensive Care Med · 2019
1.00
2
Vasopressor Therapy in the Intensive Care Unit.
PMID: 32820475
Semin Respir Crit Care Med · 2021
0.90
3
Clock gene modulates roles of OXTR and AVPR1b genes in prosociality.
PMID: 25309987
PLoS One · 2014
0.80
4
A complex selection signature at the human AVPR1B gene.
PMID: 19486526
BMC Evol Biol · 2009
0.70
5
Correlation Between Sleep Electroencephalogram, Brain-Derived Neurotrophic Factor, AVPR1B Gene Polymorphism, and Suicidal Behavior in Patients with Depression.
PMID: 36367618
Appl Biochem Biotechnol · 2023
0.60