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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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ING4
inhibitor of growth family member 4
Chromosome 12 · 12p13.31
NCBI Gene: 51147Ensembl: ENSG00000111653.21HGNC: HGNC:19423UniProt: Q9UNL4
130PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Tumor Suppressor
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
histone H4K16 acetyltransferase activityregulation of cell cycle G2/M phase transitionhistone H3K14 acetyltransferase activityhistone H4K5 acetyltransferase activityprostate cancerneoplasmFamilial prostate cancerbreast cancer
✦AI Summary

ING4 (inhibitor of growth family member 4) functions as a multifaceted tumor suppressor through epigenetic and transcriptional mechanisms. As a component of HBO1 histone acetyltransferase complexes, ING4 mediates acetylation of histone H3 at lysine-14 (H3K14ac) and functions as an epigenetic reader of H3K4me3 histone marks, regulating chr12 structure and facilitating DNA replication 12. Through these chr12 modifications, ING4 modulates transcription of genes controlling cell proliferation and apoptosis 34. ING4 suppresses multiple hallmark cancer processes: pathologic cell cycle arrest, apoptosis, autophagy, contact inhibition, and hypoxic adaptation 5. It specifically inhibits tumor angiogenesis by suppressing Sp1 expression and downstream pro-angiogenic genes (MMP-2, COX-2) 6, and represses HIF activity through interaction with prolyl hydroxylase EGLN1 7. ING4 also cooperates with p53 to enhance acetylation and transcriptional activity of p53, amplifying apoptotic responses 8. Clinically, ING4 is frequently downregulated or deleted across multiple cancer types including colorectal, breast, gastric, and hepatocellular carcinomas 695. Reduced ING4 expression correlates with lymph node metastasis, advanced disease, and poor prognosis, making it a valuable prognostic biomarker 62. ING4 restoration via gene therapy shows promising antitumor efficacy, particularly when combined with other tumor suppressors 108.

Sources cited
1
As a component of HBO1 histone acetyltransferase complexes, ING4 mediates acetylation of histone H3 at lysine-14 (H3K14ac) and functions as an epigenetic reader of H3K4me3 histone marks, regulating chr12 structure and facilitating DNA replication .
PMID: 16387653
2
As a component of HBO1 histone acetyltransferase complexes, ING4 mediates acetylation of histone H3 at lysine-14 (H3K14ac) and functions as an epigenetic reader of H3K4me3 histone marks, regulating chr12 structure and facilitating DNA replication .
PMID: 34353439
3
Through these chr12 modifications, ING4 modulates transcription of genes controlling cell proliferation and apoptosis .
PMID: 15251430
4
Through these chr12 modifications, ING4 modulates transcription of genes controlling cell proliferation and apoptosis .
PMID: 15528276
5
ING4 suppresses multiple hallmark cancer processes: pathologic cell cycle arrest, apoptosis, autophagy, contact inhibition, and hypoxic adaptation .
PMID: 30643005
6
It specifically inhibits tumor angiogenesis by suppressing Sp1 expression and downstream pro-angiogenic genes (MMP-2, COX-2) , and represses HIF activity through interaction with prolyl hydroxylase EGLN1 .
PMID: 27806345
7
It specifically inhibits tumor angiogenesis by suppressing Sp1 expression and downstream pro-angiogenic genes (MMP-2, COX-2) , and represses HIF activity through interaction with prolyl hydroxylase EGLN1 .
PMID: 15897452
8
ING4 also cooperates with p53 to enhance acetylation and transcriptional activity of p53, amplifying apoptotic responses .
PMID: 26530780
9
Clinically, ING4 is frequently downregulated or deleted across multiple cancer types including colorectal, breast, gastric, and hepatocellular carcinomas .
PMID: 19479822
10
ING4 restoration via gene therapy shows promising antitumor efficacy, particularly when combined with other tumor suppressors .
PMID: 28925992
Disease Associationsⓘ20
prostate cancerOpen Targets
0.12Weak
neoplasmOpen Targets
0.11Weak
Familial prostate cancerOpen Targets
0.11Weak
breast cancerOpen Targets
0.11Weak
hepatocellular carcinomaOpen Targets
0.10Suggestive
colorectal carcinomaOpen Targets
0.09Suggestive
melanomaOpen Targets
0.09Suggestive
osteosarcomaOpen Targets
0.08Suggestive
renal cell carcinomaOpen Targets
0.08Suggestive
gastric cancerOpen Targets
0.08Suggestive
breast neoplasmOpen Targets
0.08Suggestive
non-small cell lung carcinomaOpen Targets
0.06Suggestive
leukemiaOpen Targets
0.06Suggestive
idiopathic pulmonary fibrosisOpen Targets
0.05Suggestive
oral squamous cell carcinomaOpen Targets
0.05Suggestive
Abnormality of the skeletal systemOpen Targets
0.04Suggestive
pulmonary fibrosisOpen Targets
0.04Suggestive
cancerOpen Targets
0.04Suggestive
gliomaOpen Targets
0.04Suggestive
laryngeal neoplasmOpen Targets
0.04Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
BRPF3Protein interaction100%H3-3BProtein interaction100%H3C13Protein interaction100%EP300Protein interaction100%H3-5Protein interaction100%H3C3Protein interaction99%
Tissue Expression6 tissues
Ovary
100%
Brain
82%
Heart
81%
Liver
77%
Lung
61%
Bone Marrow
41%
Gene Interaction Network
Click a node to explore
ING4BRPF3H3-3BH3C13EP300H3-5H3C3
PROTEIN STRUCTURE
Preparing viewer…
PDB2VNF · 1.76 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
1.06LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.74 [0.53–1.06]
RankingsWhere ING4 stands among ~20K protein-coding genes
  • #3,594of 20,598
    Most Researched130 · top quartile
  • #10,649of 17,882
    Most Constrained (LOEUF)1.06
Genes detectedING4
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
The essential role of tumor suppressor gene
PMID: 30643005
Biosci Rep · 2019
1.00
2
ING4 suppresses tumor angiogenesis and functions as a prognostic marker in human colorectal cancer.
PMID: 27806345
Oncotarget · 2016
0.90
3
Roles of the tumor suppressor inhibitor of growth family member 4 (ING4) in cancer.
PMID: 34353439
Adv Cancer Res · 2021
0.80
4
Efficacy of combining ING4 and TRAIL genes in cancer-targeting gene virotherapy strategy: first evidence in preclinical hepatocellular carcinoma.
PMID: 28925992
Gene Ther · 2018
0.70
5
Multifunctional acyltransferase HBO1: a key regulatory factor for cellular functions.
PMID: 39543485
Cell Mol Biol Lett · 2024
0.60