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25 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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MAPKAPK2
MAPK activated protein kinase 2
Chromosome 1 · 1q32.1
NCBI Gene: 9261Ensembl: ENSG00000162889.12HGNC: HGNC:6887UniProt: P49137
194PubMed Papers
20Diseases
1Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Highly ConstrainedKinase
RESEARCH IMPACT
Trending
CLINICAL
Early Pipeline
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
vascular endothelial growth factor receptor signaling pathway3'-UTR-mediated mRNA stabilizationcytoplasmextracellular exosomeneurodegenerative diseaseneuroinflammatory disordermigraine disorderlysosomal storage disease
✦AI Summary

MAPKAPK2 (MK2) is a stress-activated serine/threonine kinase downstream of p38 MAPK that functions as a master regulator of post-transcriptional gene expression and cellular stress responses. Upon p38 activation, MAPKAPK2 phosphorylates multiple substrates including RNA-binding proteins (ELAVL1, HNRNPA0, PABPC1, TTP/ZFP36, ZFP36L1) to regulate transcript stability and translation of inflammatory cytokines, particularly TNF and IL6 12. During DNA damage, MAPKAPK2 translocates to the cytoplasm and phosphorylates HNRNPA0 and PARN, stabilizing GADD45A mRNA to activate checkpoint control 3. The kinase also regulates HSP27 phosphorylation, affecting its chaperone function and oxidative stress protection. Dysregulation of MAPKAPK2 has significant pathological implications: elevated expression correlates with poor prognosis and tumor progression in colorectal and head and neck cancers, where it promotes cell invasion and metastasis through MMP-2 activation 456. In hepatocellular carcinoma, MAPKAPK2 stabilization by COPS5 confers sorafenib resistance by activating ferroptosis-repressor HSPB1 7. Additionally, mTOR-regulated MAPKAPK2 translation controls the senescence-associated secretory phenotype, linking the kinase to aging and immune responses 8. These findings establish MAPKAPK2 as a therapeutic target across multiple cancer types and stress-related pathologies.

Sources cited
1
MAPKAPK2 operates post-transcriptionally to regulate TNF biosynthesis and also phosphorylates TNF receptor interactor RIPK1, providing a dual role in TNF signaling
PMID: 29275999
2
MAPKAPK2 functions as master regulator of RNA-binding proteins to control transcript stability and is implicated in tumor progression
PMID: 30850014
3
p38 MAPK and MAPKAPK2 form a positive feedback loop with unfolded protein response components (ATF4, IRE1α) during ischemic stress in glioblastoma
PMID: 39805854
4
MAPKAPK2 and its substrate HSP27 are necessary for TGF-beta-mediated MMP-2 activation and cell invasion in prostate cancer
PMID: 16407830
5
MAPKAPK2 inhibition suppresses colorectal cancer growth and invasion, with higher MAPKAPK2 levels associated with poor prognosis
PMID: 31575657
6
MAPKAPK2 promotes p16-negative head and neck cancer migration, invasion, and metastasis; its inhibition reduces circulating tumor cells and improves survival
PMID: 40185303
7
mTOR regulates MAPKAPK2 translation, which phosphorylates ZFP36L1 to control the senescence-associated secretory phenotype
PMID: 26280535
8
COPS5 stabilizes MAPKAPK2 through deubiquitination, activating HSPB1 to promote ferroptosis resistance and sorafenib resistance in hepatocellular carcinoma
PMID: 40198582
Disease Associationsⓘ20
neurodegenerative diseaseOpen Targets
0.53Moderate
neuroinflammatory disorderOpen Targets
0.39Weak
migraine disorderOpen Targets
0.38Weak
lysosomal storage diseaseOpen Targets
0.34Weak
glomerulonephritisOpen Targets
0.31Weak
sialolithiasisOpen Targets
0.26Weak
neoplasmOpen Targets
0.12Weak
Neurodevelopmental disorderOpen Targets
0.12Weak
head and neck squamous cell carcinomaOpen Targets
0.10Weak
glioblastomaOpen Targets
0.08Suggestive
hepatocellular carcinomaOpen Targets
0.08Suggestive
gliomaOpen Targets
0.08Suggestive
glioblastoma multiformeOpen Targets
0.08Suggestive
inflammatory bowel diseaseOpen Targets
0.08Suggestive
diabetes mellitusOpen Targets
0.08Suggestive
type 2 diabetes mellitusOpen Targets
0.08Suggestive
urinary bladder carcinomaOpen Targets
0.08Suggestive
Miyoshi myopathyOpen Targets
0.08Suggestive
myocardial infarctionOpen Targets
0.08Suggestive
primitive neuroectodermal tumorOpen Targets
0.07Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets1
AT-13148Phase I
MAP kinase-activated protein kinase 2 inhibitor
Related Genes
ZFP36L1Protein interaction100%HSPB1Protein interaction100%CDC25BProtein interaction98%HSPB2Protein interaction98%MAPK13Protein interaction98%MAP2K6Protein interaction98%
Tissue Expression6 tissues
Heart
100%
Bone Marrow
66%
Lung
63%
Liver
33%
Ovary
24%
Brain
21%
Gene Interaction Network
Click a node to explore
MAPKAPK2ZFP36L1HSPB1CDC25BHSPB2MAPK13MAP2K6
PROTEIN STRUCTURE
Preparing viewer…
PDB2OKR · 2.00 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.30Highly Constrained
pLIⓘ
1.00Intolerant
Observed/Expected LoF0.17 [0.10–0.30]
RankingsWhere MAPKAPK2 stands among ~20K protein-coding genes
  • #2,203of 20,598
    Most Researched194 · top quartile
  • #1,174of 17,882
    Most Constrained (LOEUF)0.30 · top 10%
Genes detectedMAPKAPK2
Sources retrieved25 papers
Response time—
📄 Sources
25▼
1
mTOR regulates MAPKAPK2 translation to control the senescence-associated secretory phenotype.
PMID: 26280535
Nat Cell Biol · 2015
1.00
2
COPS5 Triggers Ferroptosis Defense by Stabilizing MK2 in Hepatocellular Carcinoma.
PMID: 40198582
Adv Sci (Weinh) · 2025
0.90
3
MK2-TNF-Signaling Comes Full Circle.
PMID: 29275999
Trends Biochem Sci · 2018
0.80
4
MAPKAPK2: the master regulator of RNA-binding proteins modulates transcript stability and tumor progression.
PMID: 30850014
J Exp Clin Cancer Res · 2019
0.70
5
Exosomal miR-4645-5p from hypoxic bone marrow mesenchymal stem cells facilitates diabetic wound healing by restoring keratinocyte autophagy.
PMID: 38250706
Burns Trauma · 2024
0.68