HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
PRKD3
protein kinase D3
Chromosome 2 · 2p22.2
NCBI Gene: 23683Ensembl: ENSG00000115825.12HGNC: HGNC:9408UniProt: O94806
91PubMed Papers
20Diseases
5Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
Kinase
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingcytosolkinase activityplasma membraneacute myeloid leukemiasystemic mastocytosismast-cell leukemiaMastocytosis
✦AI Summary

PRKD3 (protein kinase D3) is a serine/threonine kinase that plays multifaceted roles in cellular signaling and disease pathogenesis. The protein functions as an oncogenic driver in multiple cancer types, particularly breast and gastric cancers, where it promotes tumor cell proliferation, migration, and metabolic reprogramming 123. Mechanistically, PRKD3 activates key signaling pathways including ERK1/c-MYC in breast cancer and p65/PFKFB3-mediated glycolysis in gastric cancer 32. The kinase also regulates cell cycle progression through modulation of proteins like CDK1, CyclinB1, and CHK1 4. Beyond cancer, PRKD3 serves protective functions in liver homeostasis, where its deficiency promotes hepatic fibrosis through altered macrophage polarization and sustained STAT6 activation via decreased SH2-containing protein tyrosine phosphatase-1 activity 5. Genetic studies have implicated PRKD3 variants in cardiovascular disease risk, identifying it as a potential therapeutic target for heart failure prevention 6. Additionally, PRKD3 variants are associated with Alzheimer's disease risk 7. The protein's diverse functions across different tissues suggest context-dependent roles in maintaining cellular homeostasis versus promoting pathological processes.

Sources cited
1
PRKD3 functions as an oncogenic driver in invasive breast cancer and regulates phosphoproteome networks
PMID: 28656000
2
PRKD3 promotes gastric cancer through p65/PFKFB3 activation of glycolysis
PMID: 31026442
3
PRKD3 promotes breast cancer cell proliferation by activating ERK1/c-MYC axis
PMID: 31944568
4
PRKD3 affects cell cycle progression in gastric cancer through modulation of CDK1, CyclinB1, CHK1 and PLK1
PMID: 40131654
5
PKD3 deficiency promotes liver fibrosis through macrophage polarization and STAT6 activation
PMID: 32048304
6
PRKD3 identified as potential therapeutic target for heart failure prevention
PMID: 37429843
7
PRKD3 variants associated with Alzheimer's disease risk
PMID: 34099642
Disease Associationsⓘ20
acute myeloid leukemiaOpen Targets
0.54Moderate
systemic mastocytosisOpen Targets
0.48Moderate
mast-cell leukemiaOpen Targets
0.47Moderate
MastocytosisOpen Targets
0.46Moderate
neurodegenerative diseaseOpen Targets
0.44Moderate
neoplasmOpen Targets
0.41Moderate
hypertensionOpen Targets
0.37Weak
acute myeloid leukemia by FAB classificationOpen Targets
0.37Weak
schizophreniaOpen Targets
0.34Weak
essential hypertensionOpen Targets
0.33Weak
eosinophilic esophagitisOpen Targets
0.28Weak
Alzheimer diseaseOpen Targets
0.24Weak
atrial fibrillationOpen Targets
0.23Weak
response to xenobiotic stimulusOpen Targets
0.21Weak
myelodysplastic syndromeOpen Targets
0.19Weak
kidney transplantOpen Targets
0.11Weak
prostate cancerOpen Targets
0.10Weak
oral squamous cell carcinomaOpen Targets
0.10Suggestive
breast cancerOpen Targets
0.10Suggestive
COVID-19Open Targets
0.09Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets5
CEP-2563Phase I
Protein kinase C (PKC) inhibitor
GSK-690693Phase I
Protein kinase C (PKC) inhibitor
MIDOSTAURINApproved
Tyrosine-protein kinase receptor FLT3 inhibitor
mast-cell leukemia
SOTRASTAURINPhase II
Protein kinase C (PKC) inhibitor
kidney transplant
UCN-01Phase II
3-phosphoinositide dependent protein kinase-1 inhibitor
non-small cell lung carcinoma
Related Genes
PRKCAProtein interaction98%PRKCBProtein interaction95%ITGB1Protein interaction93%RAP1AProtein interaction91%ITGALProtein interaction90%ITGAMProtein interaction90%
Tissue Expression6 tissues
Lung
100%
Ovary
90%
Brain
85%
Heart
80%
Bone Marrow
74%
Liver
47%
Gene Interaction Network
Click a node to explore
PRKD3PRKCAPRKCBITGB1RAP1AITGALITGAM
PROTEIN STRUCTURE
Preparing viewer…
PDB2D9Z · NMR
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.68LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF0.52 [0.41–0.68]
RankingsWhere PRKD3 stands among ~20K protein-coding genes
  • #5,264of 20,598
    Most Researched91
  • #956of 1,025
    FDA-Approved Drug Targets1
  • #5,082of 17,882
    Most Constrained (LOEUF)0.68
Genes detectedPRKD3
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Genome-wide association analysis and Mendelian randomization proteomics identify drug targets for heart failure.
PMID: 37429843
Nat Commun · 2023
1.00
2
Common variants in Alzheimer's disease and risk stratification by polygenic risk scores.
PMID: 34099642
Nat Commun · 2021
0.90
3
Oncogenic Protein Kinase D3 Regulating Networks in Invasive Breast Cancer.
PMID: 28656000
Int J Biol Sci · 2017
0.80
4
Protein kinase D3 promotes gastric cancer development through p65/6-phosphofructo-2-kinase/fructose-2,6-biphosphatase 3 activation of glycolysis.
PMID: 31026442
Exp Cell Res · 2019
0.70
5
CircPRKD3-loaded exosomes concomitantly elicit tumor growth inhibition and glioblastoma microenvironment remodeling via inhibiting STAT3 signaling.
PMID: 39868921
Neuro Oncol · 2025
0.60