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10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
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HDAC10
histone deacetylase 10
Chromosome 22 · 22q13.33
NCBI Gene: 83933Ensembl: ENSG00000100429.19HGNC: HGNC:18128UniProt: Q969S8
53PubMed Papers
20Diseases
12Drugs
0Pathogenic Variants
FUNCTIONAL ROLE
DNA RepairHomologous Recombination
CLINICAL
FDA Approved Target
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein lysine deacetylase activityhistone deacetylase activityprotein bindingpolyamine deacetylationneoplasmmultiple myelomaDuchenne muscular dystrophyunspecified peripheral T-cell lymphoma
✦AI Summary

HDAC10 is a class IIb histone deacetylase with dual enzymatic functions, though its primary physiological role remains incompletely characterized. Unlike most HDACs, HDAC10 functions predominantly as a polyamine deacetylase, exhibiting high specificity for N8-acetylspermidine deacetylation while showing attenuated activity toward other acetylated polyamines 1. Although histone deacetylase activity has been demonstrated in vitro, the physiological relevance of this protein-deacetylating function remains unclear 1. Mechanistically, HDAC10 employs a zinc-activated water molecule for catalysis within a sterically constrained active site that enforces substrate specificity 1. Recent studies reveal HDAC10 directly deacetylates NLRP3 at the K496 residue, switching it from acetylation to ubiquitination-mediated proteasomal degradation, thereby inhibiting NLRP3 inflammasome activation 2. Additionally, HDAC10 controls MYC-dependent transcriptional induction of the DNA polymerase POLD1, maintaining DNA replication processivity and genome integrity in lymphoid cells 3. Clinically, HDAC10 inhibition shows therapeutic potential in cancer treatment. Tucidinostat, a selective HDAC10 inhibitor, has been approved in Asia for multiple carcinomas including cervical cancer, T-cell lymphoma, and breast cancer 4. HDAC10 also plays roles in autophagy promotion and mismatch repair, with emerging recognition as a biomarker for cancer therapeutics 1.

Sources cited
1
HDAC10 is a highly specific N8-acetylspermidine deacetylase; catalyzes via zinc-activated water with sterically constrained active site; histone deacetylase activity in vitro with unclear physiological relevance; emerging biomarker for cancer treatment
PMID: 29533602
2
HDAC10 directly deacetylates NLRP3 at K496, switching acetylation to ubiquitination, inhibiting NLRP3 inflammasome and attenuating acute inflammatory diseases
PMID: 39707387
3
HDAC10 controls MYC-dependent transcriptional induction of DNA polymerase POLD1, maintaining DNA replication processivity and genome integrity in lymphoid malignancies
PMID: 40301616
4
Tucidinostat, a selective HDAC10 inhibitor (also targets HDAC1, HDAC2, HDAC3), approved in China and Japan for cervical cancer, T-cell lymphoma, brain cancer, and breast cancer
PMID: 37560925
5
HDAC10 is a polyamine deacetylase (not a lysine deacetylase); substrate specificity for N8-acetylspermidine hydrolysis; emerging target for cancer chemotherapy with selective inhibitor design strategies
PMID: 38530703
Disease Associationsⓘ20
neoplasmOpen Targets
0.55Moderate
multiple myelomaOpen Targets
0.55Moderate
Duchenne muscular dystrophyOpen Targets
0.52Moderate
unspecified peripheral T-cell lymphomaOpen Targets
0.52Moderate
Cutaneous T-cell lymphomaOpen Targets
0.49Moderate
T-cell non-Hodgkin lymphomaOpen Targets
0.46Moderate
mature T-cell and NK-cell non-Hodgkin lymphomaOpen Targets
0.45Moderate
renal cell carcinomaOpen Targets
0.37Weak
breast cancerOpen Targets
0.35Weak
lymphomaOpen Targets
0.35Weak
acute myeloid leukemiaOpen Targets
0.30Weak
myelodysplastic syndromeOpen Targets
0.29Weak
Hodgkins lymphomaOpen Targets
0.29Weak
follicular lymphomaOpen Targets
0.29Weak
polycythemia veraOpen Targets
0.28Weak
angioimmunoblastic T-cell lymphomaOpen Targets
0.26Weak
type 2 diabetes mellitusOpen Targets
0.26Weak
Abnormality of the skeletal systemOpen Targets
0.20Weak
non-small cell lung carcinomaOpen Targets
0.13Weak
melanomaOpen Targets
0.13Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Drug Targets12
ABEXINOSTATPhase III
Histone deacetylase inhibitor
follicular lymphoma
BELINOSTATApproved
Histone deacetylase inhibitor
T-cell non-Hodgkin lymphoma
CUDC-101Phase I
Epidermal growth factor receptor erbB1 inhibitor
ENTINOSTATApproved
Histone deacetylase inhibitor
neoplasm
FIMEPINOSTATPhase II
Histone deacetylase inhibitor
lymphoma
GIVINOSTATApproved
Histone deacetylase inhibitor
Duchenne muscular dystrophy
GIVINOSTAT HYDROCHLORIDEApproved
Histone deacetylase inhibitor
Duchenne muscular dystrophy
PANOBINOSTATApproved
Histone deacetylase inhibitor
multiple myeloma
PANOBINOSTAT LACTATEApproved
Histone deacetylase inhibitor
multiple myeloma
QUISINOSTATPhase II
Histone deacetylase inhibitor
ROMIDEPSINApproved
Histone deacetylase inhibitor
T-cell non-Hodgkin lymphoma
TACEDINALINEPhase II
Histone deacetylase inhibitor
Related Genes
NCOR1Protein interaction100%EP300Protein interaction97%KAT2BProtein interaction96%KAT2AProtein interaction94%H3C12Protein interaction92%H3C13Protein interaction91%
Tissue Expression6 tissues
Liver
100%
Ovary
90%
Lung
80%
Bone Marrow
22%
Brain
14%
Heart
9%
Gene Interaction Network
Click a node to explore
HDAC10NCOR1EP300KAT2BKAT2AH3C12H3C13
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q969S8
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
1.30LoF Tolerant
pLIⓘ
0.00Tolerant
Observed/Expected LoF1.09 [0.92–1.30]
RankingsWhere HDAC10 stands among ~20K protein-coding genes
  • #8,436of 20,598
    Most Researched53
  • #237of 1,025
    FDA-Approved Drug Targets7 · top quartile
  • #13,711of 17,882
    Most Constrained (LOEUF)1.30
Genes detectedHDAC10
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Recent histone deacetylase inhibitors in cancer therapy.
PMID: 37560925
Cancer · 2023
1.00
2
Epigenetic regulation of melanogenesis.
PMID: 33984527
Ageing Res Rev · 2021
0.90
3
Polyamine Deacetylase Structure and Catalysis: Prokaryotic Acetylpolyamine Amidohydrolase and Eukaryotic HDAC10.
PMID: 29533602
Biochemistry · 2018
0.80
4
Mechanism exploration and model construction for small cell transformation in EGFR-mutant lung adenocarcinomas.
PMID: 39353908
Signal Transduct Target Ther · 2024
0.70
5
HDAC10 switches NLRP3 modification from acetylation to ubiquitination and attenuates acute inflammatory diseases.
PMID: 39707387
Cell Commun Signal · 2024
0.60