HomeAboutRankingsData Sources
© 2026 GeneE
🧬
GeneE
10 sources retrieved · Most recent: April 2026 · Index updated 15 days ago
ⓘGeneE is for informational purposes only. It is not a substitute for professional medical advice, diagnosis, or treatment.
SIKE1
suppressor of IKBKE 1
Chromosome 1 · 1p13.2
NCBI Gene: 80143Ensembl: ENSG00000052723.13HGNC: HGNC:26119UniProt: Q9BRV8
31PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingprotein kinase bindingprotein-macromolecule adaptor activitysmall GTPase bindingsevere acute respiratory syndromeskull disordercardiac hypertrophygastric cancer
✦AI Summary

SIKE1 (Suppressor of IKBKE 1) functions as a physiological suppressor of IKKε and TBK1 kinases, playing critical inhibitory roles in multiple cellular pathways 1. In innate immunity, SIKE1 inhibits virus- and TLR3-triggered IRF3 activation by disrupting interactions between IKBKE/TBK1 and key signaling proteins including TICAM1/TRIF, IRF3, and RIGI, thereby suppressing interferon-stimulated response elements and IFN-β promoter activation 1. SIKE1 associates with the STRIPAK complex, forming the extended (SIKE1:SLMAP)STRIPAK complex that dephosphorylates STK3, leading to Hippo signaling inhibition and control of cell growth 2. In cardiac physiology, SIKE1 serves as an essential negative regulator of pathological cardiac hypertrophy through direct interaction with TBK1, inhibiting the TBK1-AKT signaling pathway 3. The protein also modulates DNA double-strand break repair and genomic stability, with STRIPAK-mediated MST1/2 inactivation increasing DNA repair capacity and conferring resistance to radio- and chemotherapy 4. SIKE1 expression has prognostic significance in various cancers, with elevated expression generally correlating with unfavorable outcomes in gastric cancer 5. The protein forms homo-oligomeric complexes with a primarily helical structure and exhibits dynamic conformational properties that accommodate interactions with multiple binding partners 6.

Sources cited
1
SIKE1 inhibits virus- and TLR3-triggered IRF3 activation and interferon signaling
PMID: 16281057
2
SIKE1 associates with STRIPAK complex and regulates Hippo signaling
PMID: 30622739
3
SIKE1 regulates pathological cardiac hypertrophy through TBK1-AKT pathway inhibition
PMID: 27249321
4
SIKE1-STRIPAK complex modulates DNA repair and chemotherapy resistance
PMID: 35290241
5
SIKE1 expression has prognostic significance in gastric cancer
PMID: 30487159
6
SIKE1 has helical structure and forms homo-oligomeric complexes with dynamic properties
PMID: 31074891
Disease Associationsⓘ20
severe acute respiratory syndromeOpen Targets
0.37Weak
skull disorderOpen Targets
0.32Weak
cardiac hypertrophyOpen Targets
0.07Suggestive
gastric cancerOpen Targets
0.02Suggestive
non-alcoholic steatohepatitisOpen Targets
0.02Suggestive
heart failureOpen Targets
0.01Suggestive
psoriasisOpen Targets
0.01Suggestive
dilated cardiomyopathyOpen Targets
0.01Suggestive
hypertrophic cardiomyopathyOpen Targets
0.01Suggestive
ischemiaOpen Targets
0.01Suggestive
meningococcal infectionOpen Targets
0.00Suggestive
type 1 diabetes mellitusOpen Targets
0.00Suggestive
cancerOpen Targets
0.00Suggestive
glaucomaOpen Targets
0.00Suggestive
obesityOpen Targets
0.00Suggestive
viral diseaseOpen Targets
0.00Suggestive
cryohydrocytosisOpen Targets
0.00Suggestive
diffuse large B-cell lymphomaOpen Targets
0.00Suggestive
immune system diseaseOpen Targets
0.00Suggestive
hepatocellular carcinomaOpen Targets
0.00Suggestive
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
IRF3Protein interaction100%PPP2CAProtein interaction100%STK24Protein interaction100%STK25Protein interaction100%PDCD10Protein interaction100%FGFR1OP2Protein interaction100%
Tissue Expression6 tissues
Bone Marrow
100%
Heart
89%
Liver
89%
Brain
75%
Ovary
59%
Lung
54%
Gene Interaction Network
Click a node to explore
SIKE1IRF3PPP2CASTK24STK25PDCD10FGFR1OP2
PROTEIN STRUCTURE
Preparing viewer…
PDB6AKK · 1.50 Å · X-ray
View on RCSB ↗
Constraintⓘ
LOEUFⓘ
0.55Moderately Constrained
pLIⓘ
0.94Intolerant
Observed/Expected LoF0.24 [0.12–0.55]
RankingsWhere SIKE1 stands among ~20K protein-coding genes
  • #11,799of 20,598
    Most Researched31
  • #3,477of 17,882
    Most Constrained (LOEUF)0.55 · top quartile
Genes detectedSIKE1
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Combinatorial targeting of Hippo-STRIPAK and PARP elicits synthetic lethality in gastrointestinal cancers.
PMID: 35290241
J Clin Invest · 2022
1.00
2
Pan-Cancer Analysis on the Oncogenic Role of Programmed Cell Death 10.
PMID: 36276268
J Oncol · 2022
0.90
3
LINC00665 sponges miR-641 to promote the progression of breast cancer by targeting the SNF2-related CREBBP activator protein (SRCAP).
PMID: 35152838
Bioengineered · 2022
0.80
4
miR-146a-5p circuitry uncouples cell proliferation and migration, but not differentiation, in human mesenchymal stem cells.
PMID: 23963696
Nucleic Acids Res · 2013
0.70
5
Predicting and validating a model of suppressor of IKKepsilon through biophysical characterization.
PMID: 31074891
Protein Sci · 2019
0.60