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10 sources retrieved · Most recent: April 2026 · Index updated 14 days ago
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DKK2
dickkopf Wnt signaling pathway inhibitor 2
Chromosome 4 · 4q25
NCBI Gene: 27123Ensembl: ENSG00000155011.10HGNC: HGNC:2892UniProt: Q9UBU2
55PubMed Papers
20Diseases
0Drugs
0Pathogenic Variants
DATA QUALITY
✓ Experimental GO Evidence✓ Swiss-Prot Reviewed
protein bindingnegative regulation of canonical Wnt signaling pathwaypositive regulation of canonical Wnt signaling pathwayGO:0005615androgenetic alopeciaalopeciaAbnormal nasolacrimal system morphologyintestinal obstruction
✦AI Summary

DKK2 is a secreted protein that functions as a canonical Wnt signaling inhibitor by forming complexes with LRP5/6 receptors and promoting their internalization 1. In cancer contexts, DKK2 exhibits complex roles: it promotes colorectal cancer progression by accelerating aerobic glycolysis and stimulating VEGF-independent angiogenesis through lactate production 2. Additionally, DKK2 can function as a tumor suppressor in some contexts, where its inhibition by bacterial metabolites leads to enhanced Wnt/β-catenin signaling and increased cancer cell proliferation 3. The protein also modulates immune responses, with NAT10-mediated DKK2 mRNA stabilization leading to CD8+ T cell dysfunction through cholesterol accumulation 4. In neurological contexts, DKK2 is upregulated in activated microglia during neurodegeneration and can block dendritic spine formation, contributing to synaptic dysfunction 5. During development, DKK2 serves as an arterial endothelial cell marker, indicating its role in vascular specification 6. In stroke pathology, elevated DKK2 levels correlate with worse outcomes by impairing neurovascular Wnt signaling and blood-brain barrier integrity 1. The protein's expression is regulated by epigenetic mechanisms including DNA methylation and histone modifications 73.

Sources cited
1
DKK2 promotes colorectal cancer angiogenesis through aerobic glycolysis and lactate production
PMID: 30867812
2
DKK2 serves as a marker for arterial endothelial cells during vascular development
PMID: 38348657
3
DKK2 functions as a Wnt signaling inhibitor and worsens stroke outcomes by affecting blood-brain barrier integrity
PMID: 41451773
4
DKK2 is overexpressed in activated response microglia associated with Alzheimer's disease
PMID: 31018141
5
DKK2 expression is regulated by DNA methylation in colorectal cancer
PMID: 33909798
6
DKK2 can function as a tumor suppressor whose inhibition promotes Wnt/β-catenin signaling
PMID: 40340623
7
DKK2 impairs CD8+ T cell function through cholesterol accumulation via LRP6/AKT-mTOR signaling
PMID: 41542770
8
DKK2 is upregulated in disease-associated microglia and blocks dendritic spine formation
PMID: 36599670
Disease Associationsⓘ20
androgenetic alopeciaOpen Targets
0.44Moderate
alopeciaOpen Targets
0.37Weak
Abnormal nasolacrimal system morphologyOpen Targets
0.32Weak
intestinal obstructionOpen Targets
0.32Weak
AnxietyOpen Targets
0.32Weak
cesarean sectionOpen Targets
0.31Weak
benign prostatic hyperplasiaOpen Targets
0.31Weak
HyperhidrosisOpen Targets
0.30Weak
asthmaOpen Targets
0.21Weak
respiratory tract infectious disorderOpen Targets
0.19Weak
poisoningOpen Targets
0.17Weak
VitiligoOpen Targets
0.16Weak
multiple sclerosisOpen Targets
0.15Weak
neoplasmOpen Targets
0.11Weak
benign neoplasm of eyeOpen Targets
0.11Weak
placenta praeviaOpen Targets
0.11Weak
complicationOpen Targets
0.11Weak
medical procedureOpen Targets
0.11Weak
trauma complicationOpen Targets
0.11Weak
response to stimulusOpen Targets
0.10Weak
Pathogenic Variants
No pathogenic variants reported on ClinVar for this gene.
View on ClinVar ↗
Related Genes
KREMEN1Protein interaction98%WNT3AProtein interaction95%WNT4Protein interaction95%WNT5BProtein interaction92%FRZBProtein interaction91%WNT16Protein interaction91%
Tissue Expression6 tissues
Lung
100%
Heart
74%
Brain
30%
Ovary
26%
Liver
2%
Bone Marrow
0%
Gene Interaction Network
Click a node to explore
DKK2KREMEN1WNT3AWNT4WNT5BFRZBWNT16
PROTEIN STRUCTURE
Preparing viewer…
AlphaFoldAI-predicted · UniProt Q9UBU2
View on AlphaFold ↗
Constraintⓘ
LOEUFⓘ
0.62LoF Tolerant
pLIⓘ
0.61Intermediate
Observed/Expected LoF0.37 [0.23–0.62]
RankingsWhere DKK2 stands among ~20K protein-coding genes
  • #8,190of 20,598
    Most Researched55
  • #4,354of 17,882
    Most Constrained (LOEUF)0.62 · top quartile
Genes detectedDKK2
Sources retrieved10 papers
Response time—
📄 Sources
10▼
1
Tumor-secreted dickkopf2 accelerates aerobic glycolysis and promotes angiogenesis in colorectal cancer.
PMID: 30867812
Theranostics · 2019
1.00
2
Molecular and Spatial Signatures of Mouse Embryonic Endothelial Cells at Single-Cell Resolution.
PMID: 38348657
Circ Res · 2024
0.90
3
Dickkopf-related protein 2 impairs neurovascular Wnt signalling and worsens stroke outcome.
PMID: 41451773
Eur Heart J · 2025
0.80
4
The Major Risk Factors for Alzheimer's Disease: Age, Sex, and Genes Modulate the Microglia Response to Aβ Plaques.
PMID: 31018141
Cell Rep · 2019
0.70
5
RNAM EXPRESSION AND DNA METHYLATION OF DKK2 GENE IN COLORECTAL CÂNCER.
PMID: 33909798
Arq Gastroenterol · 2021
0.60